HK Primary Care — Drug Class & MOA Reference by Condition

For FM finals / MRCGP-level recall. Generic names only — check local HA formulary for actual first-line agent/availability. Doses omitted here (ask if you want a specific one) — focus is class + mechanism.


1. Hypertension

Class Example drugs MOA
ACE inhibitor lisinopril, ramipril, perindopril Inhibit ACE → ↓angiotensin II, ↓aldosterone; ↑bradykinin (→ dry cough)
ARB losartan, valsartan, irbesartan Block AT1 receptor directly; no bradykinin effect → less cough
CCB (dihydropyridine) amlodipine, nifedipine Block L-type Ca²⁺ channels in vascular smooth muscle → vasodilation
CCB (non-dihydropyridine) diltiazem, verapamil As above + slow AV conduction/↓contractility (avoid with beta-blocker)
Thiazide/thiazide-like diuretic hydrochlorothiazide, indapamide Inhibit Na⁺-Cl⁻ cotransporter in DCT → natriuresis
Beta-blocker bisoprolol, atenolol Block β1 → ↓HR, ↓contractility, ↓renin release

NICE-style stepwise: ACEi/ARB first if <55 and non-Black African/Caribbean; CCB first if ≥55 or Black African/Caribbean origin.

2. Lipid disorder

Class Example drugs MOA
Statin atorvastatin, rosuvastatin, simvastatin Competitively inhibit HMG-CoA reductase (rate-limiting step in cholesterol synthesis) → ↑hepatic LDL receptor expression
Cholesterol absorption inhibitor ezetimibe Inhibits NPC1L1 transporter at intestinal brush border → ↓cholesterol absorption
Fibrate fenofibrate, gemfibrozil PPAR-α agonist → ↑lipoprotein lipase activity → ↓triglycerides mainly
PCSK9 inhibitor evolocumab, alirocumab Monoclonal Ab vs PCSK9 → prevents LDL-receptor degradation → ↑LDL clearance
Bile acid sequestrant cholestyramine Binds bile acids in gut, ↑hepatic conversion of cholesterol to bile acids

3. Diabetes mellitus (T2DM)

Class Example drugs MOA
Biguanide metformin Activates AMPK → ↓hepatic gluconeogenesis, ↑peripheral insulin sensitivity; no hypoglycaemia alone
Sulfonylurea gliclazide, glimepiride Bind SUR1 on pancreatic β-cell KATP channel → closure → depolarisation → insulin release
DPP-4 inhibitor (“gliptin”) sitagliptin, linagliptin Inhibit DPP-4 → ↑endogenous incretins (GLP-1/GIP) → glucose-dependent insulin release
SGLT2 inhibitor (“flozin”) empagliflozin, dapagliflozin Inhibit SGLT2 in PCT → ↓glucose reabsorption → glucosuria; also cardio/renal-protective
GLP-1 receptor agonist liraglutide, semaglutide GLP-1 agonism → ↑glucose-dependent insulin, ↓glucagon, ↓gastric emptying, central satiety
Thiazolidinedione pioglitazone PPAR-γ agonist → ↑insulin sensitivity in adipose/muscle/liver
Insulin various (basal/bolus) Direct replacement

4. URTI (incl. influenza, tonsillitis)

Class Example drugs MOA
Neuraminidase inhibitor oseltamivir Inhibits viral neuraminidase → prevents progeny virion release from infected cells (influenza only)
Penicillin phenoxymethylpenicillin (Pen V), amoxicillin β-lactam → inhibits transpeptidase (PBP) → blocks bacterial cell wall synthesis (for confirmed/high-probability GAS tonsillitis)
Antipyretic/analgesic paracetamol, ibuprofen See OA/analgesia section

Plain common cold: no antibiotics indicated — see prior summary doc.

5. Dermatitis (contact/allergic/atopic)

Class Example drugs MOA
Topical corticosteroid hydrocortisone (mild) → betamethasone (potent) Bind glucocorticoid receptor → ↓inflammatory gene transcription, ↓cytokines
Topical calcineurin inhibitor tacrolimus, pimecrolimus Inhibit calcineurin → ↓IL-2 transcription → ↓T-cell activation (steroid-sparing, good for face/eyelids)
Oral antihistamine (H1) cetirizine, chlorphenamine H1 receptor antagonism → ↓itch/wheal-flare
Emollient various Barrier repair, ↓transepidermal water loss (foundation of all eczema management)

6. Gastroenteritis

Class Example drugs MOA
Oral rehydration salts ORS Na⁺/glucose co-transport drives water absorption in gut
5-HT3 antagonist ondansetron Blocks 5-HT3 receptors centrally (CTZ) and peripherally (vagal afferents) → antiemetic
Dopamine antagonist (prokinetic) metoclopramide D2 antagonism (crosses BBB → EPS risk) + 5-HT4 agonism → prokinetic/antiemetic
Opioid receptor agonist (gut) loperamide μ-opioid agonism in gut wall, minimal CNS penetration → ↓peristalsis (avoid if bloody/febrile diarrhoea)
Fluoroquinolone (selected cases) ciprofloxacin Inhibits bacterial DNA gyrase/topoisomerase IV (for specific bacterial/traveller’s diarrhoea only)

7. Allergic rhinitis

Class Example drugs MOA
Intranasal corticosteroid fluticasone, mometasone Local anti-inflammatory — first-line for moderate-severe/persistent Sx
2nd-gen oral antihistamine cetirizine, loratadine, fexofenadine Peripheral H1 antagonism, minimal sedation
Leukotriene receptor antagonist montelukast CysLT1 receptor antagonist → ↓leukotriene-mediated inflammation
Intranasal antihistamine azelastine Local H1 antagonism
Mast cell stabiliser sodium cromoglicate Inhibits mast cell degranulation

8. Dyspepsia / GERD

Class Example drugs MOA
PPI omeprazole, esomeprazole, lansoprazole Irreversibly inhibit H⁺/K⁺-ATPase (proton pump) on gastric parietal cells
H2 receptor antagonist famotidine Blocks H2 receptors on parietal cells → ↓acid secretion (less potent than PPI)
Antacid aluminium/magnesium hydroxide Direct acid neutralisation
Prokinetic domperidone Peripheral D2 antagonist (limited BBB crossing → less EPS than metoclopramide)
H. pylori eradication PPI + amoxicillin + clarithromycin (metronidazole if penicillin-allergic) Triple therapy — acid suppression + dual antibiotic

9. Obesity

Class Example drugs MOA
Lipase inhibitor orlistat Inhibits pancreatic/gastric lipase → ↓dietary fat absorption
GLP-1 receptor agonist (higher dose) liraglutide (Saxenda), semaglutide (Wegovy) As above — also central appetite suppression

10. OA knee / knee complaints

Class Example drugs MOA
Paracetamol Mechanism incompletely understood; central COX inhibition/other CNS effects — first-line analgesic
Topical NSAID diclofenac gel Local COX-1/2 inhibition → ↓prostaglandin synthesis, less systemic exposure
Oral NSAID (non-selective) ibuprofen, naproxen Non-selective COX-1/2 inhibition
Oral NSAID (COX-2 selective) celecoxib Selective COX-2 inhibition → less GI toxicity, ↑cardiovascular risk
Intra-articular corticosteroid triamcinolone, methylprednisolone Local anti-inflammatory injection

11. Gout

Class Example drugs MOA
NSAID (acute) naproxen, indomethacin COX inhibition
Colchicine (acute) colchicine Binds tubulin → inhibits microtubule polymerisation → ↓neutrophil chemotaxis/degranulation
Corticosteroid (acute, if NSAID/colchicine CI) prednisolone (oral) or intra-articular Anti-inflammatory
Xanthine oxidase inhibitor (chronic ULT) allopurinol, febuxostat Inhibit xanthine oxidase → ↓uric acid production
Uricosuric (chronic ULT) probenecid Inhibits renal tubular urate reabsorption → ↑excretion

Don’t start urate-lowering therapy during an acute flare; continue if already established.

12. Depressive disorder

Class Example drugs MOA
SSRI sertraline, fluoxetine, escitalopram Inhibit serotonin reuptake transporter (SERT) → ↑synaptic 5-HT
SNRI venlafaxine, duloxetine Inhibit both SERT and NET → ↑5-HT and noradrenaline
NaSSA mirtazapine α2-antagonist (↑NA/5-HT release) + 5-HT2/5-HT3 antagonist — sedating, appetite-stimulating
TCA amitriptyline Inhibit NA/5-HT reuptake; also anticholinergic/antihistaminic (more SEs, used at low dose for pain too)

13. Thyroid disorder

Class Example drugs MOA
Thyroid hormone replacement levothyroxine (T4) Synthetic T4, peripherally converted to active T3
Thionamide (antithyroid) carbimazole (prodrug → methimazole) Inhibits thyroid peroxidase → blocks iodination/coupling of thyroglobulin
Thionamide (antithyroid) propylthiouracil (PTU) As above + inhibits peripheral T4→T3 conversion; preferred 1st trimester pregnancy (less teratogenic, but hepatotoxicity risk)
Beta-blocker (symptom control) propranolol Non-selective β-blockade → controls tremor/palpitations/tachycardia in thyrotoxicosis

14. Ischaemic heart disease

Class Example drugs MOA
Antiplatelet (COX inhibitor) aspirin Irreversible COX-1 inhibition → ↓thromboxane A2 → ↓platelet aggregation
Antiplatelet (P2Y12 inhibitor) clopidogrel, ticagrelor Block ADP-mediated P2Y12 receptor → ↓platelet activation
Beta-blocker bisoprolol, metoprolol ↓HR/contractility → ↓myocardial O2 demand
Statin atorvastatin As above — also plaque stabilisation
Nitrate GTN (sublingual/spray), isosorbide mononitrate NO donor → venodilation (↓preload) + coronary vasodilation
ACE inhibitor ramipril Cardioprotective remodelling, esp. post-MI/LV dysfunction

15. Low back pain

Class Example drugs MOA
Paracetamol / NSAID as above As above — first-line
Muscle relaxant (short-term, selected cases) diazepam (limited use) GABA-A positive allosteric modulation

Avoid routine opioids for chronic non-specific LBP; exercise/physio is mainstay.

16. Benign prostatic hyperplasia (BPH)

Class Example drugs MOA
α1-blocker tamsulosin, doxazosin Selective α1A antagonism → relaxes prostatic/bladder neck smooth muscle (fast symptom relief)
5α-reductase inhibitor finasteride, dutasteride Inhibit conversion testosterone→DHT → shrinks prostate over months (slower onset, reduces long-term progression)

17. Dermatophytosis (tinea)

Class Example drugs MOA
Allylamine (topical/oral) terbinafine Inhibits squalene epoxidase → squalene accumulation (toxic) + ergosterol deficiency
Azole (topical) clotrimazole, miconazole Inhibit lanosterol 14α-demethylase (CYP450 enzyme) → blocks ergosterol synthesis
Azole (oral, extensive/nail/scalp disease) itraconazole, fluconazole As above, systemic

18. Constipation

Class Example drugs MOA
Bulk-forming ispaghula husk (psyllium) ↑stool bulk/water retention → mechanical peristaltic stimulus
Osmotic lactulose, macrogol (PEG) Non-absorbable → draws water into lumen osmotically (lactulose also fermented → mild acidification)
Stimulant senna, bisacodyl Stimulate enteric nerves/colonic motility directly
Stool softener docusate sodium Surfactant — allows water/fat to penetrate stool

19. Urinary tract infection

Class Example drugs MOA
Nitrofuran nitrofurantoin Bacterial nitroreductases generate reactive intermediates → damage DNA/ribosomal proteins (multi-target); avoid near-term pregnancy & significant renal impairment
Folate synthesis inhibitor trimethoprim Inhibits bacterial dihydrofolate reductase
Phosphonic acid derivative fosfomycin Inhibits MurA enzyme → blocks peptidoglycan (cell wall) synthesis; single-dose regimen
β-lactam/β-lactamase inhibitor co-amoxiclav For resistant/complicated cases

20. Cerebrovascular disease (stroke/TIA secondary prevention)

Class Example drugs MOA
Antiplatelet aspirin, clopidogrel As above
Statin (high-intensity) atorvastatin As above
DOAC (if AF-related) apixaban, rivaroxaban (direct Xa inhibitors); dabigatran (direct thrombin inhibitor) Direct inhibition of clotting factor Xa or IIa
Vitamin K antagonist warfarin Inhibits vitamin K epoxide reductase → ↓synthesis of factors II, VII, IX, X

21. Vertigo / dizziness

Class Example drugs MOA
Histamine analogue betahistine Weak H1 agonist + H3 antagonist → ↑inner ear blood flow (used in Ménière’s)
Dopamine antagonist (acute vertigo/vomiting) prochlorperazine D2 antagonism at CTZ + vestibular sedation
Antihistamine (vestibular sedative) cinnarizine H1 antagonism + mild Ca²⁺ channel blockade

22. Asthma

Class Example drugs MOA
SABA (reliever) salbutamol β2-agonism → bronchodilation
ICS (preventer) beclometasone, budesonide, fluticasone Local anti-inflammatory — reduces airway inflammation/hyperresponsiveness
LABA salmeterol, formoterol Longer-acting β2-agonism — always combined with ICS, never alone
LTRA montelukast CysLT1 antagonist
LAMA (add-on, severe) tiotropium Muscarinic (M3) antagonism → bronchodilation
Anti-IgE (severe allergic asthma) omalizumab Monoclonal Ab binds free IgE → prevents mast cell/basophil activation

23. Bursitis / tendinitis / synovitis

Class Example drugs MOA
NSAID (oral/topical) as above As above
Corticosteroid injection triamcinolone Local anti-inflammatory

24. Liver disease

Class Example drugs MOA
Nucleos(t)ide analogue (chronic Hep B) tenofovir, entecavir Inhibit HBV reverse transcriptase/DNA polymerase
Aldosterone antagonist (ascites) spironolactone Mineralocorticoid receptor antagonism → K⁺-sparing diuresis
Osmotic laxative (hepatic encephalopathy) lactulose Traps ammonia as ammonium in gut lumen (acidification) + laxative effect → ↓ammonia absorption
Non-selective beta-blocker (variceal prophylaxis) propranolol ↓cardiac output (β1) + splanchnic vasoconstriction (unopposed α, β2 blockade) → ↓portal pressure

25. Abdominal pain (functional/IBS-type)

Class Example drugs MOA
Antimuscarinic antispasmodic hyoscine butylbromide Antimuscarinic → relaxes GI smooth muscle; poor oral bioavailability (mainly peripheral effect)
Musculotropic antispasmodic mebeverine Direct smooth muscle relaxant, minimal anticholinergic effect

26. Neck / shoulder pain

Same as low back pain — paracetamol/NSAIDs first-line; consider topical NSAID for localised tendinopathy.

27. Anxiety

Class Example drugs MOA
SSRI/SNRI as above First-line for GAD (same as depression)
Benzodiazepine (short-term only) diazepam, lorazepam Positive allosteric modulator at GABA-A receptor → ↑Cl⁻ conductance; risk of dependence, avoid long-term
5-HT1A partial agonist buspirone Non-sedating, non-addictive alternative, slower onset
Beta-blocker (somatic/performance anxiety) propranolol β-blockade → controls tremor/palpitations, no effect on psychological Sx

28. Headache

Class Example drugs MOA
Simple analgesic (tension-type) paracetamol, NSAIDs As above
Triptan (migraine, acute) sumatriptan 5-HT1B/1D agonism → cranial vasoconstriction + inhibits trigeminal neuropeptide (CGRP) release
Migraine prophylaxis propranolol, topiramate, amitriptyline (low dose) Propranolol: β-blockade; Topiramate: multiple (Na⁺ channel block, ↑GABA, ↓glutamate); Amitriptyline: as above

Watch for medication-overuse headache with frequent analgesic/triptan use.

29. Sleep disturbance

Class Example drugs MOA
Z-drug zolpidem, zopiclone GABA-A receptor agonism (non-benzodiazepine site) — short-term use only
Melatonin melatonin MT1/MT2 receptor agonism — circadian regulation, useful in elderly

CBT-I is first-line; pharmacotherapy is short-term adjunct only.

30. Eye complaints (blepharitis, stye, chalazion, red eye)

Class Example drugs MOA
Topical antibiotic chloramphenicol drops/ointment Inhibits bacterial 50S ribosomal subunit → blocks protein synthesis (for bacterial conjunctivitis/infective blepharitis)
Topical antihistamine/mast cell stabiliser olopatadine, sodium cromoglicate For allergic conjunctivitis
Warm compress + lid hygiene Mainstay for blepharitis/stye/chalazion; antibiotics only if cellulitis/spreading infection

31. Osteoporosis

Class Example drugs MOA
Bisphosphonate alendronate, zoledronic acid Bind hydroxyapatite, taken up by osteoclasts → inhibit farnesyl pyrophosphate synthase → osteoclast apoptosis
RANKL inhibitor denosumab Monoclonal Ab vs RANKL → prevents osteoclast differentiation/activation
PTH analogue (anabolic, severe cases) teriparatide Intermittent PTH(1-34) exposure → net osteoblast stimulation (anabolic, unlike continuous PTH)
SERM raloxifene Selective oestrogen receptor modulator — oestrogenic effect on bone, antagonist on breast/uterus
Adjunct calcium + vitamin D Substrate/cofactor for bone mineralisation

32. Urticaria

Class Example drugs MOA
2nd-gen antihistamine (may uptitrate to 4× dose) cetirizine, fexofenadine Peripheral H1 antagonism — first-line
Oral corticosteroid (short course, severe/acute) prednisolone Anti-inflammatory
Anti-IgE (chronic spontaneous urticaria, refractory) omalizumab As above

33. Haemorrhoids

Class Example drugs MOA
Topical corticosteroid + local anaesthetic hydrocortisone + lidocaine combo Anti-inflammatory + local analgesia (short courses only)
Bulk laxative ispaghula Softens stool, ↓straining

34. Anaemia

Class Example drugs MOA
Iron replacement ferrous sulfate, ferrous fumarate Replenishes iron stores for haem synthesis
B12 replacement hydroxocobalamin (IM), cyanocobalamin (oral) Cofactor for DNA synthesis/methylation — replacement
Folate replacement folic acid Cofactor for DNA synthesis — replacement
Erythropoiesis-stimulating agent (CKD-related) erythropoietin (epoetin alfa) Stimulates erythroid progenitor cells in bone marrow

35. Skin infections

Class Example drugs MOA
Topical antibiotic (impetigo) fusidic acid, mupirocin Fusidic acid: inhibits bacterial protein synthesis (EF-G); Mupirocin: inhibits isoleucyl-tRNA synthetase
β-lactam (cellulitis) flucloxacillin Penicillinase-resistant β-lactam — covers S. aureus/strep
Alternative (penicillin allergy/MRSA risk) clindamycin, doxycycline, co-trimoxazole Clindamycin: inhibits 50S ribosome; Doxycycline: inhibits 30S ribosome; Co-trimoxazole: dual folate synthesis blockade

36. Acute bronchitis

Mostly viral — symptomatic care only (as for URTI). Consider doxycycline/amoxicillin only if suspected bacterial superinfection, or in COPD/high-risk patients with purulent sputum + systemic upset.

37. Herpes zoster

Class Example drugs MOA
Nucleoside analogue (antiviral) aciclovir, valaciclovir, famciclovir Require viral thymidine kinase for activation → inhibit viral DNA polymerase, chain termination. Start within 72h of rash onset
Neuropathic agent (post-herpetic neuralgia) gabapentin, pregabalin, amitriptyline See neuropathic pain section below

38. Chest pain

Not a distinct drug class of its own — management follows the underlying cause (IHD #14, GERD #8). GTN may be used as both symptomatic relief and a rough diagnostic pointer toward cardiac cause (though not definitive).

39. Cough

Follows underlying cause: URTI/bronchitis (#4/#36, mostly supportive), asthma (#22, consider ICS trial if cough-variant), GERD (#8, PPI trial if reflux-associated cough).


Bonus — genuinely high-yield in HK primary care but not explicit in your list

Peripheral/diabetic neuropathy (very common given DM prevalence)

Class Example drugs MOA
Gabapentinoid gabapentin, pregabalin Bind α2δ subunit of voltage-gated Ca²⁺ channels → ↓excitatory neurotransmitter release
SNRI duloxetine As above — licensed specifically for diabetic neuropathic pain
TCA (low dose) amitriptyline As above, used off-label for neuropathic pain at lower doses than antidepressant use

Immunisation (Preventive category)

Vaccine type Examples Mechanism
Inactivated (killed) injectable influenza, Hep A Non-replicating antigen — immune response without infection risk
Live attenuated MMR, varicella, live nasal flu Weakened live organism — replicates transiently → robust/durable immunity; avoid in pregnancy/immunosuppression
Subunit/recombinant Hep B, HPV (recombinant capsid protein), recombinant zoster (Shingrix-type) Purified antigen component only
Toxoid tetanus, diphtheria Inactivated toxin — immunity against toxin, not organism
Polysaccharide/conjugate pneumococcal (PPSV23 polysaccharide vs PCV13/15/20 conjugate) Conjugate linked to carrier protein → T-cell dependent response, works in young children (polysaccharide alone is T-independent, poor in <2yo)
mRNA COVID-19 mRNA vaccines mRNA encoding viral antigen (e.g. spike protein) taken up by cells → transient antigen expression → immune response

Notes on local practice

This reflects internationally standard drug classes/mechanisms and largely NICE-consistent first-line reasoning — the pharmacology itself doesn’t change by jurisdiction. What genuinely can differ in HK: exact first-line agent per HA Drug Formulary, GOPC prescribing restrictions (some drug classes are specialist-initiated only in the public system), and availability of certain newer agents (e.g., SGLT2i/GLP-1 agonist access, PCSK9i restrictions) outside private practice. I don’t have the current HA Drug Formulary to confirm exact tier/restriction status — worth cross-checking against it directly for anything formulary-specific in an OSCE/finals context.