| Inhibitor | Summary of CDK inhibitors | ||
|---|---|---|---|
| CDKs | Diseases | References | |
| Palbociclib | CDK4/6 | metastatic breast cancer | [16-20] |
| Ribociclib | CDK4/6 | metastatic breast cancer | [22-28] |
| Abemaciclib | CDK4/6 | high risk early breast cancer | [30-33] |
| SLS009 | CDK9 | acute myeloid leukemia, peripheral T-cell lymphoma | [36, 37] |
| TP-1287 | broad-range | Ewing sarcoma | [39] |
| Alvocidib | broad-range | acute myeloid leukemia | [40] |
| NUV-422 | CDK2/CDK4/CDK6 | malignant glioma (discontinued) | [41-44] |